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BDBM50337367 4-(1H-indazol-5-yl)-2-methylthiazole::CHEMBL1682542

SMILES: Cc1nc(cs1)-c1ccc2[nH]ncc2c1

InChI Key: InChIKey=LYYSRRLDPCPRDC-UHFFFAOYSA-N

Data: 6 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50337367
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Rho-associated protein kinase 2 (Human)	BDBM50337367 (4-(1H-indazol-5-yl)-2-methylthiazole \| CHEMBL16825...) Show SMILES Show InChI	GoogleScholar	UniChem		513	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glycogen synthase kinase-3 beta (Human)	BDBM50337367 (4-(1H-indazol-5-yl)-2-methylthiazole \| CHEMBL16825...) Show SMILES Show InChI	GoogleScholar	UniChem		2.86E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase PAK 4 (Human)	BDBM50337367 (4-(1H-indazol-5-yl)-2-methylthiazole \| CHEMBL16825...) Show SMILES Show InChI	GoogleScholar	UniChem		>3.75E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Human)	BDBM50337367 (4-(1H-indazol-5-yl)-2-methylthiazole \| CHEMBL16825...) Show SMILES Show InChI	GoogleScholar	UniChem		4.16E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Aurora kinase B (Human)	BDBM50337367 (4-(1H-indazol-5-yl)-2-methylthiazole \| CHEMBL16825...) Show SMILES Show InChI	GoogleScholar	UniChem		4.45E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Human)	BDBM50337367 (4-(1H-indazol-5-yl)-2-methylthiazole \| CHEMBL16825...) Show SMILES Show InChI	GoogleScholar	UniChem		>8.88E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair