BDBM50342914 6-(1-methyl-1H-indazol-6-yl)-N-(thiophen-2-ylmethyl)quinazolin-4-amine::CHEMBL1397997

SMILES Cn1ncc2ccc(cc12)-c1ccc2ncnc(NCc3cccs3)c2c1

InChI Key InChIKey=UDDOADGLWVILSJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50342914   

TargetDual specificity protein kinase CLK4(Human)
National Human Genome Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342914BDBM50342914(6-(1-methyl-1H-indazol-6-yl)-N-(thiophen-2-ylmethy...)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of Clk4 kinase using ATP as substrate by 33P radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
National Human Genome Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50342914BDBM50342914(6-(1-methyl-1H-indazol-6-yl)-N-(thiophen-2-ylmethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Dyrk1A kinase using ATP as substrate by 33P radiolabeled kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed