BDBM50400774 CHEMBL2204983

SMILES CC1(CC1)OC(=O)N1CCC(CC1)n1ncc(COc2ccc(cc2)-n2cnnn2)c1C#N

InChI Key InChIKey=SDGHYCIXEZKBLQ-UHFFFAOYSA-N

Data  1 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50400774   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400774(CHEMBL2204983)
Affinity DataKi:  30nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400774(CHEMBL2204983)
Affinity DataEC50:  22nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400774(CHEMBL2204983)
Affinity DataEC50:  15nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed