BDBM50430603 CHEMBL2338735

SMILES CCC[C@](C)(O)[C@H]1C[C@]23CC[C@]1(OC)[C@@H]1Oc4c5c(C[C@H]2N(CC2CC2)CC[C@@]315)ccc4O

InChI Key InChIKey=UOKRJODYISPCKA-DPJBPYIISA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50430603   

TargetMu-type opioid receptor(GUINEA PIG)
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50430603(CHEMBL2338735)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DAMGO from MOR in Hartley guinea pig membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50430603(CHEMBL2338735)
Affinity DataKi:  2nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50430603(CHEMBL2338735)
Affinity DataIC50:  0.490nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed