BDBM534170 6-Cyclopropyl-4-(dimethylamino)-N-[(2-methyl-8-quinolyl)sulfonyl]benzofuran-2-carboxamide::WO2022081842, Example 43

SMILES CN(C)c1cc(cc2oc(cc12)C(=O)NS(=O)(=O)c1cccc2ccc(C)nc12)C1CC1

InChI Key InChIKey=QSSZPSCTOYDGGS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 534170   

TargetHistone acetyltransferase KAT6A [507-778](Homo sapiens)
The Broad Institute

WIPO
LigandPNGBDBM534170(6-Cyclopropyl-4-(dimethylamino)-N-[(2-methyl-8-qui...)
Affinity DataIC50:  13nMAssay Description: Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed