TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 0.245nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 0.309nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human erythrocytes AChE using acetylthiocholine iodide as substrate measured after 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of human erythrocytes AChE using acetylthiocholine iodide as substrate measured after 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 372nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Instituto De Investigaciones Biol£Gicas Clemente Estable
Curated by ChEMBL
Affinity DataIC50: 457nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 4.54E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 6.95E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 9.79E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Universidad Nacional De C£Rdoba
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human erythrocytes AChE using acetylthiocholine iodide as substrate measured after 30 mins by Ellman's methodMore data for this Ligand-Target Pair