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Found 22 with Last Name = 'amparo' and Initial = 'ec'
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50451005(CHEMBL290376 | DuP-714)
Affinity DataKi:  0.0420nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076548(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-3-(2-h...)
Affinity DataKi:  7nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076545(CHEMBL422722 | {1-[2-(4-Benzyl-piperidin-1-yl)-2-o...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50451005(CHEMBL290376 | DuP-714)
Affinity DataKi:  9nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076540(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-1H-ind...)
Affinity DataKi:  18nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076549(CHEMBL366643 | {1-[2-(4-Benzyl-piperidin-1-yl)-2-o...)
Affinity DataKi:  19nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076547(1-{2-[4-(2-Fluoro-benzyl)-piperidin-1-yl]-2-oxo-et...)
Affinity DataKi:  24nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076538(1-{2-[4-(3-Fluoro-benzyl)-piperidin-1-yl]-2-oxo-et...)
Affinity DataKi:  24nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076537(3-{1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-5-c...)
Affinity DataKi:  28nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076545(CHEMBL422722 | {1-[2-(4-Benzyl-piperidin-1-yl)-2-o...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076546(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-1H-ind...)
Affinity DataKi:  140nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076542(6-(4-Benzyl-piperidine-1-sulfonyl)-1H-indole-3-car...)
Affinity DataKi:  210nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076537(3-{1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-5-c...)
Affinity DataKi:  280nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076539(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-1H-ben...)
Affinity DataKi:  300nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076548(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-3-(2-h...)
Affinity DataKi:  310nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076542(6-(4-Benzyl-piperidine-1-sulfonyl)-1H-indole-3-car...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076546(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-1H-ind...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076543(1-[2-(4-Benzoyl-piperidin-1-yl)-2-oxo-ethyl]-1H-in...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076540(1-[2-(4-Benzyl-piperidin-1-yl)-2-oxo-ethyl]-1H-ind...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076541(1-{2-[4-(Hydroxy-phenyl-methyl)-piperidin-1-yl]-2-...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibitory activity of the compound against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076541(1-{2-[4-(Hydroxy-phenyl-methyl)-piperidin-1-yl]-2-...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076543(1-[2-(4-Benzoyl-piperidin-1-yl)-2-oxo-ethyl]-1H-in...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibition of Coagulation factor IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed