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Found 23 with Last Name = 'andré' and Initial = 'a'
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161249(3a,11a-dihydroxy-4''-imino-9,15a-dimethyl-1-(5-oxo...)
Affinity DataIC50:  68nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161262(11a-hydroxy-3a,13a-di(hydroxymethyl)-9,15a-dimethy...)
Affinity DataIC50:  75nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161244(CHEMBL369515 | Uscharin derivative)
Affinity DataIC50:  1.89E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161268(CHEMBL366906 | Uscharin derivative)
Affinity DataIC50:  4.08E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161245(11a-hydroxy-3a-hydroxymethyl-4''-imino-9,15a-dimet...)
Affinity DataIC50:  1.21E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404744(CHEMBL19047)
Affinity DataIC50:  2.45E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404740(CHEMBL436338)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161246(11a-hydroxy-3a-hydroxymethyl-4''-imino-9,15a-dimet...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161253(CHEMBL426228 | Uscharin derivative)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161272(CHEMBL262795 | Uscharin derivative)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161252(CHEMBL427124 | Uscharin derivative)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM14363(3-(2-propoxyphenyl)-2,4,7,8,9-pentazabicyclo[4.3.0...)
Affinity DataIC50:  6.31E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404743(CHEMBL273765)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404745(CHEMBL18262)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)
Affinity DataIC50:  8.13E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404739(CHEMBL276918)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404748(CHEMBL19032 | NSC-115922)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404741(CHEMBL278972)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404746(NSC-115919 | PENTAACETYLQUERCETIN)
Affinity DataIC50:  2.75E+5nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404742(CHEMBL18487)
Affinity DataIC50:  3.50E+5nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404747(CHEMBL18415)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010981((Ro 20-1724)4-(3-Butoxy-4-methoxy-benzyl)-imidazol...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404738(CHEMBL18609)
Affinity DataIC50:  1.30E+6nMAssay Description:Inhibition of rat brain particulate cGMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed