Affinity DataKi: 5nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 142nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 331nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 345nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 390nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 656nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 690nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 810nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 925nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 945nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.68E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.21E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Ability to inhibit the binding of [125I]-C5a anaphylatoxin chemotactic receptor to polymorphonuclear leukocyte (PMNL) membrane receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.69E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibitory activity against [125I]-rC5a binding to C5a anaphylatoxin chemotactic receptor in human polymorphonuclear leukocyte (PMNL) membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.05E+4nMAssay Description:In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranesMore data for this Ligand-Target Pair