TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Irreversible inhibition of rat hormone sensitive lipase assessed as relative residual activity by kinetic analysisMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Irreversible inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of human AChE assessed as equilibrium binding by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+3nMAssay Description:Inhibition of equine BChE assessed as equilibrium constant using butyrylthiocholine iodide as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8.90E+3nMAssay Description:Inhibition of human AChE assessed as equilibrium constant using acetylthiocholine as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of human AChE assessed as equilibrium binding by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.60E+4nMAssay Description:Inhibition of human AChE assessed as equilibrium binding by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+5nMAssay Description:Inhibition of human AChE assessed as equilibrium binding by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+5nMAssay Description:Inhibition of human AChE assessed as equilibrium binding by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Inhibition of housefly CSMA AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human BChE using butyrylthiocholine as substrate measured for 30 secs by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human AChE using p-nitrophenyl acetate as substrate measured for 30 secs by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 30 min followed by substrate addition measured ever...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of horse BChE using butyrylthiocholine iodide as substrate measured for 30 secs by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate measured for 30 secs by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human AChE at pH 6More data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human AChE at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 30 min followed by substrate addition measured ever...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human AChE by modified Ellman's spectrophotometric methodMore data for this Ligand-Target Pair
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of rat hormone sensitive lipase assessed as oleic acid release from [3H]triolein by scintillation countingMore data for this Ligand-Target Pair