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Found 629 with Last Name = 'isik' and Initial = 's'
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428850(CHEMBL2337539)
Affinity DataKi:  0.330nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428841(CHEMBL2337134)
Affinity DataKi:  0.530nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428844(CHEMBL2337544)
Affinity DataKi:  0.570nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428843(CHEMBL2337132)
Affinity DataKi:  0.590nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428845(CHEMBL1594453)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428850(CHEMBL2337539)
Affinity DataKi:  0.640nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428838(CHEMBL2337530)
Affinity DataKi:  0.650nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428837(CHEMBL2337531)
Affinity DataKi:  0.650nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428846(CHEMBL2337543)
Affinity DataKi:  0.660nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428837(CHEMBL2337531)
Affinity DataKi:  0.670nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428842(CHEMBL2337133)
Affinity DataKi:  0.670nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428849(CHEMBL2337540)
Affinity DataKi:  0.670nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428847(CHEMBL2337542)
Affinity DataKi:  0.720nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067987(CHEMBL3400811)
Affinity DataKi:  0.760nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428844(CHEMBL2337544)
Affinity DataKi:  0.860nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428848(CHEMBL2337541)
Affinity DataKi:  0.860nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50304157(3-(2-Thienyl)-2-thiocarbamoyl-2,3,4,5,6,7-hexahydr...)
Affinity DataKi:  0.900nMAssay Description:Competitive inhibition of MAOB in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067992(CHEMBL3400816)
Affinity DataKi:  0.910nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067994(CHEMBL3400798)
Affinity DataKi:  0.910nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067948(CHEMBL3400804)
Affinity DataKi:  0.920nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428836(CHEMBL2337532)
Affinity DataKi:  0.930nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428846(CHEMBL2337543)
Affinity DataKi:  0.930nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50304152(3-(2-Furyl)-2-thiocarbamoyl-2,3,4,5,6,7-hexahydro-...)
Affinity DataKi:  0.960nMAssay Description:Competitive inhibition of MAOB in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428842(CHEMBL2337133)
Affinity DataKi:  0.960nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067995(CHEMBL3400799)
Affinity DataKi:  0.970nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067987(CHEMBL3400811)
Affinity DataKi:  0.970nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Balikesir University

Curated by ChEMBL
LigandPNGBDBM10870(2-N-(4-aminobenzene)-1,3,4-thiadiazole-2,5-disulfo...)
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428838(CHEMBL2337530)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428840(CHEMBL2337528)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428835(CHEMBL2337533)
Affinity DataKi:  2.40nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067996(CHEMBL3400800)
Affinity DataKi:  2.60nMAssay Description:Inhibition of human recombinant carbonic anhydrase 9 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Balikesir University

Curated by ChEMBL
LigandPNGBDBM50428833(CHEMBL2337534)
Affinity DataKi:  2.70nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Balikesir University

Curated by ChEMBL
LigandPNGBDBM10885((4R)-4-(ethylamino)-2-(3-methoxypropyl)-1,1-dioxo-...)
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant CA2 by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428836(CHEMBL2337532)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428830(CHEMBL2337537)
Affinity DataKi:  3.5nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428833(CHEMBL2337534)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067992(CHEMBL3400816)
Affinity DataKi:  3.90nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Balikesir University

Curated by ChEMBL
LigandPNGBDBM50428838(CHEMBL2337530)
Affinity DataKi:  4.20nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM50304156(3-(2-Furyl)-2-(N-phenyllthiocarbamoyl)-3,3a,4,5,6,...)
Affinity DataKi:  4.22nMAssay Description:Competitive inhibition of MAOA in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428834(CHEMBL1347917)
Affinity DataKi:  4.30nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50067996(CHEMBL3400800)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human recombinant carbonic anhydrase 12 expressed in Escherichia coli pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428835(CHEMBL2337533)
Affinity DataKi:  4.90nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428839(CHEMBL2337529)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428849(CHEMBL2337540)
Affinity DataKi:  5.20nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428833(CHEMBL2337534)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Balikesir University

Curated by ChEMBL
LigandPNGBDBM50428846(CHEMBL2337543)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50428839(CHEMBL2337529)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Balikesir University

Curated by ChEMBL
LigandPNGBDBM50428834(CHEMBL1347917)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Hacettepe University

Curated by ChEMBL
LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataKi:  5.53nMAssay Description:Competitive inhibition of MAOA in rat liver homogenate by spectrophotometricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
Salman Bin Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human recombinant carbonic anhydrase-12-mediated CO2 hydration preincubated for 10 mins by stopped-flow assayMore data for this Ligand-Target Pair
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