Affinity DataKi: 3nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Vernalis (R&D)
Curated by ChEMBL
Vernalis (R&D)
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity towards human Dopamine receptor D2 (long) by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Vernalis (R&D)
Curated by ChEMBL
Vernalis (R&D)
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Inhibition of fluorescein-labelled VER160364 binding to PDHK1 (unknown origin) after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Vernalis (R&D)
Curated by ChEMBL
Vernalis (R&D)
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Inhibition of fluorescein-labelled VER160364 binding to PDHK1 (unknown origin) after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of fluorescein-labelled VER160364 from HSP90A (unknown origin) after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Vernalis (R&D)
Curated by ChEMBL
Vernalis (R&D)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of fluorescein-labelled VER160364 binding to PDHK1 (unknown origin) after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Vernalis (R&D)
Curated by ChEMBL
Vernalis (R&D)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter (DAT) of cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Vernalis (R&D)
Curated by ChEMBL
Vernalis (R&D)
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Inhibition of fluorescein-labelled VER160364 binding to PDHK1 (unknown origin) after 90 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair