Affinity DataKi: 89nMAssay Description:Displacement of [3H]meselurgine from human recombinant 5HT2C receptor expressed in Swiss mouse 3T3 cells by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Displacement of [3H]meselurgine from human recombinant 5HT2C receptor expressed in Swiss mouse 3T3 cells by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 424nMAssay Description:Displacement of [3H]meselurgine from human recombinant 5HT2C receptor expressed in Swiss mouse 3T3 cells by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 728nMAssay Description:Displacement of [3H]meselurgine from human recombinant 5HT2C receptor expressed in Swiss mouse 3T3 cells by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 970nMAssay Description:Binding affinity to rat 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human alpha2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to human muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to rat alpha1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]meselurgine from human recombinant 5HT2C receptor expressed in Swiss mouse 3T3 cells by SPAMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of dofetilide from hERGMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of rat NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of rabbit NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMpH: 7.0Assay Description:Inhibition of human kidney NEP at pH 7More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMpH: 7.0Assay Description:Inhibition of human kidney NEP at pH 7More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMpH: 7.0Assay Description:Inhibition of human kidney NEP at pH 7More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human recombinant NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMpH: 7.0Assay Description:Inhibition of human kidney NEP at pH 7More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.4Assay Description:Inhibition of human kidney NEP at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 10.2nMAssay Description:Inhibition of rabbit NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 10.2nMAssay Description:Inhibition of rabbit NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 10.5nMpH: 7.4Assay Description:Inhibition of human kidney NEP at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 12.6nMpH: 7.4Assay Description:Inhibition of human kidney NEP at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 13.8nMpH: 7.4Assay Description:Inhibition of human kidney NEP at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 14.3nMAssay Description:Inhibition of rat NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 14.3nMAssay Description:Inhibition of rat NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 18.9nMpH: 7.0Assay Description:Inhibition of human kidney NEP at pH 7More data for this Ligand-Target Pair
Affinity DataIC50: 18.9nMAssay Description:Inhibition of human NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 19.7nMAssay Description:Inhibition of human recombinant NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 19.7nMAssay Description:Inhibition of human recombinant NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 31.8nMpH: 7.4Assay Description:Inhibition of human kidney NEP at pH 7.4More data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 176nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 184nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 195nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 205nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair
Affinity DataIC50: 213nMAssay Description:Inhibition of dog NEPMore data for this Ligand-Target Pair