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Found 154 with Last Name = 'shams' and Initial = 'g'
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  0.302nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470917(CHEMBL120278)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470918(CHEMBL123596)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  2nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470916(CHEMBL121704)
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470924(CHEMBL122990)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470919(CHEMBL332964)
Affinity DataKi:  7.80nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470922(CHEMBL122992)
Affinity DataKi:  8.70nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471350(CHEMBL102763)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470920(CHEMBL121964)
Affinity DataKi:  12nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50036910(4-(1-Naphthalen-1-yl-ethyl)-1H-imidazole | CHEMBL3...)
Affinity DataKi:  13nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  21nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
Affinity DataKi:  25nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471342(CHEMBL322907)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470860(CHEMBL105328)
Affinity DataKi:  33nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  44nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  44nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  45nMAssay Description:Binding affinity against Beta-2 adrenergic receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  47nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  49nMAssay Description:Binding affinity against Beta-2 adrenergic receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50470860(CHEMBL105328)
Affinity DataKi:  55nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50470861(CHEMBL322844)
Affinity DataKi:  57nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82493(CAS_128658 | NSC_128658 | TMQ, (+/-)-8-Fluoro)
Affinity DataKi:  58nMAssay Description:Binding affinity against beta-2 adrenergic receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50471350(CHEMBL102763)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  76nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79.4nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  87nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471338(CHEMBL105347)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82493(CAS_128658 | NSC_128658 | TMQ, (+/-)-8-Fluoro)
Affinity DataKi:  98nMAssay Description:Binding affinity against beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471346(CHEMBL330185)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471343(CHEMBL319221)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470859(CHEMBL105487)
Affinity DataKi:  122nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50471343(CHEMBL319221)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  162nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50470862(CHEMBL102076)
Affinity DataKi:  165nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471347(CHEMBL319984)
Affinity DataKi:  169nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  178nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  182nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470918(CHEMBL123596)
Affinity DataKi:  186nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50471338(CHEMBL105347)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50471347(CHEMBL319984)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471348(CHEMBL103448)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50223426(CHEBI:10304 | Corbadrine | Levonordefrin | Neo-Cob...)
Affinity DataKi:  205nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM50036910(4-(1-Naphthalen-1-yl-ethyl)-1H-imidazole | CHEMBL3...)
Affinity DataKi:  224nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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