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Found 190 with Last Name = 'siddiqi' and Initial = 'mi'
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524365(CHEMBL4579211)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human H3 receptor expressed in HEK293T cells measured after 90 mins by liquid scintillat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524374(CHEMBL4453810)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant human H3 receptor expressed in HEK293T cells measured after 90 mins by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecreted chorismate mutase(Mycobacterium tuberculosis H37Rv)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50209967(4-[2-(3,4-dimethoxy-phenyl)-ethylamino]-3-nitro-5-...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of chorismate mutase in Mycobacterium tuberculosis H37Rv strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecreted chorismate mutase(Mycobacterium tuberculosis H37Rv)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50209968((Z)-2-(4-chlorophenyl)-3-(4,5-dimethoxy-2-nitrophe...)
Affinity DataKi:  1.77E+4nMAssay Description:Inhibition of chorismate mutase in Mycobacterium tuberculosis H37Rv strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecreted chorismate mutase(Mycobacterium tuberculosis H37Rv)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50209969(2-(3-(tert-butoxycarbonyl)-2-phenylthiazolidine-4-...)
Affinity DataKi:  2.11E+4nMAssay Description:Inhibition of chorismate mutase in Mycobacterium tuberculosis H37Rv strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSecreted chorismate mutase(Mycobacterium tuberculosis H37Rv)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50209966(CHEMBL242816 | methyl 4-(methylamino)-3-nitrobenzo...)
Affinity DataKi:  2.88E+4nMAssay Description:Inhibition of chorismate mutase in Mycobacterium tuberculosis H37Rv strainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014498((S)-2-(4-(((2-amino-4-oxo-3,4-dihydroquinazolin-6-...)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM18771((2S)-2-[(4-{[(2-amino-4-oxo-1,4-dihydroquinazolin-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50006689((S)-2-(2-fluoro-4-(((2-methyl-4-oxo-3,4-dihydroqui...)
Affinity DataIC50:  20nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014496((S)-2-(2-fluoro-4-(((2-methoxy-4-oxo-3,4-dihydroqu...)
Affinity DataIC50:  36nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524380(CHEMBL4451233)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50012036((S)-2-(5-(((2-methyl-4-oxo-3,4-dihydroquinazolin-6...)
Affinity DataIC50:  40nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50006687((S)-2-(4-(((2-methyl-4-oxo-3,4-dihydroquinazolin-6...)
Affinity DataIC50:  40nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524380(CHEMBL4451233)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014501((S)-2-(2-fluoro-4-((2-fluoroethyl)((2-methyl-4-oxo...)
Affinity DataIC50:  43nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014506((S)-2-(4-(ethyl((2-methyl-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50:  45nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524379(CHEMBL4540275)
Affinity DataIC50: <50nMAssay Description:Displacement of [I125]bolton hunter-CCK-8S from recombinant human CCK1 receptor expressed in stable CHO cells measured after 1 to 2 hrs by microscint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014494((S)-2-(2-fluoro-4-(((4-oxo-3,4-dihydroquinazolin-6...)
Affinity DataIC50:  58nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014497((S)-2-(2-fluoro-4-(((2-(hydroxymethyl)-4-oxo-3,4-d...)
Affinity DataIC50:  58nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524368(CHEMBL4452406)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014495((S)-2-(4-(((2-methoxy-4-oxo-3,4-dihydroquinazolin-...)
Affinity DataIC50:  68nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014518((S)-2-(2-methoxy-4-(((2-methyl-4-oxo-3,4-dihydroqu...)
Affinity DataIC50:  68nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524368(CHEMBL4452406)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014514((S)-2-(2-chloro-4-(((2-methyl-4-oxo-3,4-dihydroqui...)
Affinity DataIC50:  74nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014516((S)-2-(4-(allyl((2-methyl-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50:  76nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014505((S)-2-(2-fluoro-4-((2-hydroxyethyl)((2-methyl-4-ox...)
Affinity DataIC50:  78nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524367(CHEMBL4580450)
Affinity DataIC50:  85nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014527((S)-2-(2-hydroxy-4-(((2-methyl-4-oxo-3,4-dihydroqu...)
Affinity DataIC50:  89nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524367(CHEMBL4580450)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014485((S)-2-(4-(((2-(hydroxymethyl)-4-oxo-3,4-dihydroqui...)
Affinity DataIC50:  98nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50006694((S)-2-(2-fluoro-4-(methyl((2-methyl-4-oxo-3,4-dihy...)
Affinity DataIC50:  120nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014517((S)-2-(2-chloro-4-(ethyl((2-methyl-4-oxo-3,4-dihyd...)
Affinity DataIC50:  120nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50005353(CHEMBL320464)
Affinity DataIC50:  129nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014476((S)-2-(4-(((2-ethyl-4-oxo-3,4-dihydroquinazolin-6-...)
Affinity DataIC50:  141nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50005352(CHEMBL101425)
Affinity DataIC50:  145nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50012044((S)-2-(5-(ethyl((2-methyl-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50:  151nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50012038((S)-2-(5-((2-fluoroethyl)((2-methyl-4-oxo-3,4-dihy...)
Affinity DataIC50:  158nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014504((S)-2-(4-((cyanomethyl)((2-methyl-4-oxo-3,4-dihydr...)
Affinity DataIC50:  170nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50012045((S)-2-(4-(ethyl((2-methyl-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50:  170nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014480((S)-2-(4-(((4-oxo-3,4-dihydroquinazolin-6-yl)methy...)
Affinity DataIC50:  170nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014520((S)-2-(4-(ethyl((2-methyl-4-oxo-3,4-dihydroquinazo...)
Affinity DataIC50:  191nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50415844(CHEMBL1094274)
Affinity DataIC50:  191nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014483((S)-2-(4-((2-fluoroethyl)((2-(hydroxymethyl)-4-oxo...)
Affinity DataIC50:  219nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014470((S)-2-(4-(((4-oxo-2-phenyl-3,4-dihydroquinazolin-6...)
Affinity DataIC50:  219nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50415849(CHEMBL1097599)
Affinity DataIC50:  229nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50415840(CHEMBL1095919)
Affinity DataIC50:  229nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014479((S)-2-(4-(((4-oxo-2-((pyrimidin-2-ylthio)methyl)-3...)
Affinity DataIC50:  240nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
Meerut Institute Of Engineering And Technology

Curated by ChEMBL
LigandPNGBDBM50014473((S)-2-(4-((2-fluoroethyl)((2-methyl-4-oxo-3,4-dihy...)
Affinity DataIC50:  240nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524363(CHEMBL4585616)
Affinity DataIC50:  240nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Academy Of Scientific And Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50524363(CHEMBL4585616)
Affinity DataIC50:  245nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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