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Found 145 with Last Name = 'sonders' and Initial = 'm'
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81980(Butanserin | CAS_87051-46-5 | NSC_65652)
Affinity DataKi:  1.86nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81981(7-(2-(4-(4-fluorobenzoyl)piperidino)ethyl)theophyl...)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  5.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81978(CAS_159037 | NSC_159037 | R 56413)
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81979(CAS_5051-62-7 | CAS_65636 | Fluprofylline | Guanab...)
Affinity DataKi:  28.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  72.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81980(Butanserin | CAS_87051-46-5 | NSC_65652)
Affinity DataKi:  75.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81981(7-(2-(4-(4-fluorobenzoyl)piperidino)ethyl)theophyl...)
Affinity DataKi:  120nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  191nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81979(CAS_5051-62-7 | CAS_65636 | Fluprofylline | Guanab...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81978(CAS_159037 | NSC_159037 | R 56413)
Affinity DataKi:  257nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81978(CAS_159037 | NSC_159037 | R 56413)
Affinity DataKi:  282nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataKi:  295nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81981(7-(2-(4-(4-fluorobenzoyl)piperidino)ethyl)theophyl...)
Affinity DataKi:  417nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
The Oregon Health Sciences University

Curated by PDSP Ki Database
LigandPNGBDBM81979(CAS_5051-62-7 | CAS_65636 | Fluprofylline | Guanab...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006990(CHEMBL299499 | N-Adamantan-1-yl-N'-(4-iodo-phenyl)...)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006986(CHEMBL442356 | N-Adamantan-1-yl-N'-(4-fluoro-2-met...)
Affinity DataIC50:  3.20nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010779(CHEMBL310003 | N-Bicyclo[2.2.1]hept-2-yl-N'-(2-iod...)
Affinity DataIC50:  4nMAssay Description:In vitro inhibitory activity against [3H]-DTG in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010759(CHEMBL553896 | N-Adamantan-1-yl-N'-(2-iodo-phenyl)...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010779(CHEMBL310003 | N-Bicyclo[2.2.1]hept-2-yl-N'-(2-iod...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against [3H]-DTG in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010782(CHEMBL553347 | N-Adamantan-2-yl-N'-(2-iodo-phenyl)...)
Affinity DataIC50:  5.20nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010742(CHEMBL81773 | N-Bicyclo[2.2.1]hept-2-yl-N'-o-tolyl...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010795(CHEMBL81461 | N-Adamantan-2-yl-N'-o-tolyl-guanidin...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010759(CHEMBL553896 | N-Adamantan-1-yl-N'-(2-iodo-phenyl)...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006991(CHEMBL55970 | N-Adamantan-1-yl-N'-(2-iodo-phenyl)-...)
Affinity DataIC50:  6.20nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006983(CHEMBL55873 | N-Adamantan-1-yl-N'-(4-methoxy-2-met...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006988(CHEMBL54407 | N-Adamantan-1-yl-N'-(3-methoxy-pheny...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010742(CHEMBL81773 | N-Bicyclo[2.2.1]hept-2-yl-N'-o-tolyl...)
Affinity DataIC50:  7.70nMAssay Description:In vitro inhibitory activity against [3H]-DTG in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006987(CHEMBL55769 | N-Adamantan-1-yl-N'-(3-iodo-phenyl)-...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010764(CHEMBL543597 | N-Adamantan-1-yl-N'-cyclohexyl-guan...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010756(CHEMBL81835 | N-Adamantan-1-yl-N'-o-tolyl-guanidin...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010756(CHEMBL81835 | N-Adamantan-1-yl-N'-o-tolyl-guanidin...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006993(CHEMBL293059 | N-Adamantan-1-yl-N'-(2-fluoro-pheny...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010747(CHEMBL543201 | CHEMBL78777 | N,N'-Bis-(3-ethyl-phe...)
Affinity DataIC50:  8.30nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006989(CHEMBL292450 | N-Adamantan-1-yl-N'-(4-fluoro-pheny...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006992(CHEMBL292668 | N-Adamantan-1-yl-N'-(4-methoxy-phen...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010768(CHEMBL553535 | N,N'-Di-adamantan-1-yl-guanidine; h...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010768(CHEMBL553535 | N,N'-Di-adamantan-1-yl-guanidine; h...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010766(CHEMBL79164 | N-Cyclohexyl-N'-o-tolyl-guanidine)
Affinity DataIC50:  12nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010764(CHEMBL543597 | N-Adamantan-1-yl-N'-cyclohexyl-guan...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50006984(CHEMBL413257 | N-Adamantan-1-yl-N'-(3-fluoro-pheny...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010760(CHEMBL310170 | N,N'-Bis-(2-ethyl-phenyl)-guanidine)
Affinity DataIC50:  13.8nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010758(CHEMBL312600 | N,N'-Bis-(2-iodo-phenyl)-guanidine)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010760(CHEMBL310170 | N,N'-Bis-(2-ethyl-phenyl)-guanidine)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010766(CHEMBL79164 | N-Cyclohexyl-N'-o-tolyl-guanidine)
Affinity DataIC50:  15nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010748(CHEMBL540291 | N-(3,5-Dimethyl-adamantan-1-yl)-N'-...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institutions

Curated by ChEMBL
LigandPNGBDBM50010758(CHEMBL312600 | N,N'-Bis-(2-iodo-phenyl)-guanidine)
Affinity DataIC50:  16nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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