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Found 2 Enz. Inhib. hit(s) with Target = 'Guanine nucleotide binding protein, alpha q polypeptide'
TargetGuanine nucleotide binding protein, alpha q polypeptide(Cricetulus griseus)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50514449(CHEMBL4171381)
Affinity DataIC50:  33nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGuanine nucleotide binding protein, alpha q polypeptide(Cricetulus griseus)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50468902(CHEMBL4288881)
Affinity DataIC50:  95nMAssay Description:Inhibition of Gq-mediated signalling in CHOK1 cells stably expressing M1 muscarinic receptor assessed as inhibition of carbachol-induced IP1 producti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed