TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Inhibition of Fragile histidine triad prorein hydrolytic activityMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 900nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 7.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 8.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 8.60E+4nMAssay Description:Inhibition assay using Fhit with ApppBODIPY.More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of human FHIT expressed in Escherichia coli BL21(DE3)-RIL cells using AP3A as substrate pretreated for 10 mins followed by substrate addit...More data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human FHIT assessed as reduction in AP3Aase activity measured after 45 mins by HPLC analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.73E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair
TargetBis(5'-adenosyl)-triphosphatase(Homo sapiens (Human))
Polish Academy Of Sciences
Curated by ChEMBL
Polish Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human FHIT incubated for 1hr in presence of tokyogreen-labeled CMP probe by fluorescence based analysisMore data for this Ligand-Target Pair