Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50036244
TargetNociceptin receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity against delta-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity against delta-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity against mu-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity against mu-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataKi:  33nMAssay Description:Binding affinity against kappa-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  332nMAssay Description:Binding affinity against kappa-opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038642(22-methyl-(2R,13S)-14-oxa-4,22-diazaheptacyclo[13....)
Affinity DataIC50: 920nMAssay Description:Antagonist activity against mu-opioid receptor in guinea pig ileum in the presence of morphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038642(22-methyl-(2R,13S)-14-oxa-4,22-diazaheptacyclo[13....)
Affinity DataIC50: 990nMAssay Description:Antagonist activity against kappa-opioid receptor in guinea pig ileum in the presence of ethylketazocineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038642(22-methyl-(2R,13S)-14-oxa-4,22-diazaheptacyclo[13....)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against delta-opioid receptor in mouse vas deferens in the presence of DADLEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity against kappa-opioid receptor in guinea pig ileum in the presence of ethylketazocineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50038641(22-cyclopropylmethyl-(2R,13S)-14-oxa-4,22-diazahep...)
Affinity DataIC50: 8.20E+3nMAssay Description:Antagonist activity against delta-opioid receptor in mouse vas deferens in the presence of DADLEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataIC50: 1.12E+4nMAssay Description:Antagonist activity against mu-opioid receptor in guinea pig ileum in the presence of morphineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataIC50: 4.59E+5nMAssay Description:Antagonist activity against delta-opioid receptor in mouse vas deferens in the presence of DADLEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed