Affinity DataEC50: 0.160nMAssay Description:Agonist activity at full length human ERbeta receptor assessed as transcriptional activity incubated for 22 to 24 hrs by cell based luciferase report...More data for this Ligand-Target Pair
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at full length human ERalpha receptor assessed as transcriptional activity incubated for 22 to 24 hrs by cell based luciferase repor...More data for this Ligand-Target Pair
Affinity DataEC50: 0.370nMAssay Description:Displacement of fluormone from GST-tagged ERbeta receptor LBD (unknown origin) measured after 60 mins by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >10nMAssay Description:Antagonist activity at full length human ERbeta receptor assessed as inhibition of estradiol-induced activation incubated for 22 to 24 hrs by cell ba...More data for this Ligand-Target Pair
Affinity DataEC50: >50nMAssay Description:Antagonist activity at full length human ERalpha receptor assessed as inhibition of estradiol-induced activation incubated for 22 to 24 hrs by cell b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.34E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature rabbitMore data for this Ligand-Target Pair
Affinity DataEC50: 1.68E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
Affinity DataEC50: 3.37E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in squirrel monkeyMore data for this Ligand-Target Pair
Affinity DataEC50: >3.37E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair