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Found 4 of ec50 for monomerid = 50275055
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  9.77E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed