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Compile Data Set for Download or QSAR

Found 1 hit of ki for monomerid = 301529   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Mitogen-activated protein kinase kinase kinase 12


(Homo sapiens (Human))
BDBM301529
PNG
(US10131675, Example 14)
Show SMILES CC1(C)OCCn2c1nc1c(nc(nc21)-c1cnc(N)nc1)N1CC2CCOC2C1
Show InChI InChI=1S/C20H24N8O2/c1-20(2)18-24-14-16(27-9-11-3-5-29-13(11)10-27)25-15(12-7-22-19(21)23-8-12)26-17(14)28(18)4-6-30-20/h7-8,11,13H,3-6,9-10H2,1-2H3,(H2,21,22,23)
PDB

KEGG

UniProtKB/SwissProt
UniProtKB/TrEMBL

antibodypedia
GoogleScholar
PC cid
PC sid
UniChem
US Patent
990n/an/an/an/an/an/an/an/a



Genentech Inc

US Patent


Assay Description
DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...


US Patent US10131675 (2018)


BindingDB Entry DOI: 10.7270/Q21G0P92
More data for this
Ligand-Target Pair