Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50088437
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen

LigandPNGBDBM50088437(1-(5-Phenyl-pyridin-3-yl)-[1,4]diazepane | CHEMBL3...)
Affinity DataKi:  0.800nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine-binding protein(Lymnaea stagnalis)
University Of Copenhagen

LigandPNGBDBM50088437(1-(5-Phenyl-pyridin-3-yl)-[1,4]diazepane | CHEMBL3...)
Affinity DataKi:  8.90nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen

LigandPNGBDBM50088437(1-(5-Phenyl-pyridin-3-yl)-[1,4]diazepane | CHEMBL3...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed