Found 10 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1B' and Ligand = 'BDBM50014407'
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataKi: 208nMAssay Description:The compound was tested for their binding affinity towards 5-hydroxytryptamine 1B receptor from rat striatum using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataKi: 310nMAssay Description:Ability to displace [3H]5-HT bound to 5-hydroxytryptamine 1B receptor in rat striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataKi: 310nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor of rat striatum.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataKi: 320nMAssay Description:Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataIC50: 380nMAssay Description:Inhibition of radiolabeled [3H]-5-HT ligand binding to 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataIC50: 7.08E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1B receptor was measured using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Affinity DataIC50: 7.08E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair