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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50309343'
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50309343(8-methyl-2,3,4,5,5a,6-hexahydro-[1,4]diazepino[1,7...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2C receptor expressed in HEK293E cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50309343(8-methyl-2,3,4,5,5a,6-hexahydro-[1,4]diazepino[1,7...)
Affinity DataEC50:  61nMAssay Description:Agonist activity at 5HT2C receptor in rat fundusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50309343(8-methyl-2,3,4,5,5a,6-hexahydro-[1,4]diazepino[1,7...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant 5HT2C receptor expressed in HEK293E cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed