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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50116458'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50116458(1-Methyl-2-phenyl-1,4,6,7-tetrahydro-1,3,4,5a,8-pe...)
Affinity DataKi:  500nMAssay Description:Inhibition against Adenosine A1 receptor of rat fat cell membranes (functional antagonist activity)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50116458(1-Methyl-2-phenyl-1,4,6,7-tetrahydro-1,3,4,5a,8-pe...)
Affinity DataKi:  1.83E+3nMAssay Description:Binding affinity against Adenosine A1 receptor by displacing [3H]CHA radioligand in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed