Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50149597'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Warwick

Curated by ChEMBL
LigandPNGBDBM50149597(CHEMBL3771184)
Affinity DataIC50:  0.398nMAssay Description:Agonist activity at human Adenosine A1 receptor transfected in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Warwick

Curated by ChEMBL
LigandPNGBDBM50149597(CHEMBL3771184)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at human Adenosine A1 receptor expressed in yeast cells coexpressed with chimeric GPA1/Galphai1 after 16 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed