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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50196564'
TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50196564((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(methylamino)...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50196564((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(methylamino)...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]ABMECA from adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed