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Found 3 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM82498'
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  7.41nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataEC50:  501nMAssay Description:Inhibitory activity against Beta-1 adrenergic receptor in guinea pig atria after treatment with the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed