Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]CP-55940 from rat CB1 receptor expressed in rat brain membrane by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 96nMAssay Description:Agonist activity at human CB1 receptor transfected in human U2OS cells assessed as beta-arrestin2-GFP aggregation after 40 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at human CB1 receptor transfected in HEK293 cells assessed as reduction in forskolin-stimulated cAMP accumulation after 30 minsMore data for this Ligand-Target Pair