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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50277309'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277309(3,3,3-trifluoro-2-methyl-N-(4-methyl-3-(morpholino...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CP55940 from human cloned CB2 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277309(3,3,3-trifluoro-2-methyl-N-(4-methyl-3-(morpholino...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277309(3,3,3-trifluoro-2-methyl-N-(4-methyl-3-(morpholino...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human cloned CB2 receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed