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Found 2 Enz. Inhib. hit(s) with Target = 'DNA gyrase subunit A' and Ligand = 'BDBM50117914'
TargetDNA gyrase subunit A(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Achillion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117914(1-Cyclopropyl-1,4-dihydro-6-fluoro-8-methoxy-7-(3-...)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of DNA supercoiling activity of wild type Mycobacterium tuberculosis DNA gyrase AMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50117914(1-Cyclopropyl-1,4-dihydro-6-fluoro-8-methoxy-7-(3-...)
Affinity DataIC50:  7.64E+5nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase Ser84Leu mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed