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Found 2 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM18624'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandPNGBDBM18624((18Z)-18-({3-[(1E)-1-(ethoxyimino)ethyl]thiophen-2...)
Affinity DataIC50:  0.5nM EC50:  0.400nMpH: 7.5Assay Description:GR-Mediated Agonist Activity Assay- GR-mediated activation by compounds is measured against maximal activation of dexamethasone in the same experimen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandPNGBDBM18624((18Z)-18-({3-[(1E)-1-(ethoxyimino)ethyl]thiophen-2...)
Affinity DataIC50:  0.5nM EC50:  1.90nMpH: 7.5Assay Description:GR-Mediated Antagonist Activity Assay- GR-mediated antagonist activity is measured in the presence of a concentration of dexamethasone empirically de...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed