Affinity DataKi: 320nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity against Histamine H1 receptor using receptor binding assay in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Ability to displace [3H]-pyrilamine from H1 receptor in rat brain membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition constant against histamine H1 receptorMore data for this Ligand-Target Pair