TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at human H2R-Gsalphas expressed in Sf9 cells at 0.1 nM to 10 uM by steady state GTPase activity assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataKd: 6.92E+4nMAssay Description:Compound is evaluated for histamine H2 receptor agonistic activity in guinea pig cerebral cortex using [3H]tiotidine as radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 1.17E+5nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Activity at human recombinant histamine H2 receptor-Gsalpha fusion protein expressed in Sf9 cells by steady-state GTPase activity assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.20E+3nMAssay Description:Activity at guinea pig recombinant histamine H2 receptor-Gsalpha fusion protein expressed in Sf9 cells by steady-state GTPase activity assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig spontaneously beating right atrium assessed as positive chronotropic activityMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at human histamine H2 receptor expressed in Sf9 cells coexpressing GsalphaS protein by steady-state GTPase assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at histamine H2 receptor in spontaneously beating guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at GsalphaS-fused human histamine H2 receptor expressed in Sf9 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at guinea pig H2R-Gsalphas expressed in Sf9 cells at 0.1 nM to 10 uM by steady state GTPase activity assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at GsalphaS-fused guinea pig histamine H2 receptor expressed in Sf9 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 650nMAssay Description:Agonist activity at human H2 receptor expressed in 293-EBNA cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 463nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]-tiotidineMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at H2R in spontaneously beating guinea pig right atrium assessed as increase in heart rateMore data for this Ligand-Target Pair