Affinity DataKi: 17nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Antagonist activity assessed as inhibition of U50488-stimulated [35S]GTP-gamma-S binding to human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity at cloned human kappa opioid receptor by [3H]diprenorphine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Partial agonist activity at human cloned kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity against Opioid receptor kappa 1 using [3H]-Ethylketocyclazocine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity towards kappa-opioid receptor by displacement of [3H]-EKC at from guinea pig cortical tissueMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity was determined against Opioid receptor kappa 1
using [3H]-Ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair
using [3H]-Ethylketocyclazocine as radioligandMore data for this Ligand-Target Pair