TargetMineralocorticoid receptor(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica (Iqm-Csic)
Curated by ChEMBL
Instituto De Qu£Mica M£Dica (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-Aldosterone from MR overexpressed in human 293 cells measured after 2 hrs by Microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetMineralocorticoid receptor(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica (Iqm-Csic)
Curated by ChEMBL
Instituto De Qu£Mica M£Dica (Iqm-Csic)
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human MR overexpressed in HEK293 cells assessed as inhibition of aldosterone-induced response measured after overnight incubat...More data for this Ligand-Target Pair