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Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 12' and Ligand = 'BDBM365290'
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM365290((1-Methyl-1H-imidazol- 4-yl)-{3-[2-(2-methyl- pyrr...)
Affinity DataKi:  1.72nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent