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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50006590'
TargetMuscarinic acetylcholine receptor M1(RAT)
Novo Nordisk Cns Division

Curated by ChEMBL
LigandPNGBDBM50006590(1-Methyl-5-(4-octyl-[1,2,5]thiadiazol-3-yl)-1,2,3,...)
Affinity DataIC50:  56nMAssay Description:In vitro binding affinity against Muscarinic acetylcholine receptor M1 from rat hippocampus, using [3H]-pirenzepine (Pz) as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Novo Nordisk Cns Division

Curated by ChEMBL
LigandPNGBDBM50006590(1-Methyl-5-(4-octyl-[1,2,5]thiadiazol-3-yl)-1,2,3,...)
Affinity DataIC50:  428nMAssay Description:In vitro binding affinity against Muscarinic acetylcholine receptor M1 from rat hippocampus, using [3H]-oxotremorine-M (Oxo-M) as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed