Affinity DataKi: 0.200nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]osanetant from human recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]osanetant from wild type human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards cloned human Tachykinin receptor 3 (hNK-3) expressed in CHO cells using [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding Affinity of [125I]-MePhe7-NKB towards Tachykinin receptor 3-CHO cell membranes(n=3-8)More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-SB222200 from recombinant human NK3R expressed in CHO cell membranes after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity to human NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Displacement of [3H]-SB222200 from rat NK3R after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity to rat NK3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Compound was tested for binding affinity against human Tachykinin receptor 3 in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Tachykinin receptor 3 binding affinity was determined by incubation with CHO cells expressing human NK3 receptorsMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Ability to displace [3H]senktide succinyl-[Asp9MePhe8]-SP (6-13)} from Tachykinin receptor 3 of guinea pig cerebral cortex membraneMore data for this Ligand-Target Pair
Affinity DataKd: 18.6nMAssay Description:Competitive inhibition at wild type human NK3 expressed in HEK293 cells assessed as decrease in [MePhe7]NKB-induced [3H]IP accumulation after 20 minsMore data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Binding affinity to wild type human NK3 receptor expressed in HEK293 cells assessed as [3H]IP accumulation after 45 minsMore data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Equilibrium binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.0800nMAssay Description:Apparent binding affinity to guinea pig NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.150nMAssay Description:Equilibrium binding affinity to guinea pig NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.220nMAssay Description:Apparent binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair