Found 2 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50006990'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 in human MDA-MB-468 cell membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Drexel University College Of Medicine
Curated by ChEMBL
Drexel University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair