Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50009049'
TargetSigma non-opioid intracellular receptor 1(RAT)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50009049((+/-)(1-Methyl-2-phenyl-ethyl)-(4-phenyl-butyl)-am...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity towards sigma opioid receptor was determined in rat cerebral homogenate using [3H]haloperidol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50009049((+/-)(1-Methyl-2-phenyl-ethyl)-(4-phenyl-butyl)-am...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity towards sigma opioid receptor in guinea pig cerebral homogenate using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed