Found 5 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50110577'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 699nMAssay Description:In vitro binding affinity of the compound in LLC-PK1 cells by Dopamine transporter binding assay by using [125I]-IPT as a radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Binding affinity for dopamine transporter expressed in LCK PK1 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:In vitro inhibition of [3H]-WIN- 35,428 binding to human dopamine transporter expressed in canine kidney cellsMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-GBR-12,935 binding to dopamine transporter (DAT) of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Pennsylvania
Curated by ChEMBL
University Of Pennsylvania
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:In vitro displacement of [3H]-GBR-12,935 from human dopamine transporter expressed in HEK-293 cellsMore data for this Ligand-Target Pair