Found 2 Enz. Inhib. hit(s) with Target = 'Transmembrane domain-containing protein TMIGD3' and Ligand = 'BDBM50259308'
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Universita Degli Studi Di Firenze
Curated by ChEMBL
Universita Degli Studi Di Firenze
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cell membranes after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Universita Degli Studi Di Firenze
Curated by ChEMBL
Universita Degli Studi Di Firenze
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Antagonist activity at human A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP production by [3H]cA...More data for this Ligand-Target Pair