Affinity DataKi: 3nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]DOI from cloned human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 515nMAssay Description:Inhibitory activity against 5HT4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.27E+3nMAssay Description:Displacement of [3H]clonidine from cloned human adrenergic alpha2A receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Displacement of [3H]clonidine from cloned human adrenergic Alpha-2C receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.87E+3nMAssay Description:Inhibitory activity against 5HT1D receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against SERTMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against 5HT1B receptorMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Alcon Research
Curated by ChEMBL
Alcon Research
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against NETMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against 5HT6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory activity against adrenergic alpha-1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory activity against adrenergic alpha-1A receptorMore data for this Ligand-Target Pair