TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of LCK in human Jurkat cells assessed as ZAP70 phosphorylation by FACS assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of tie2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 4.23E+3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of RetMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Her1More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Her2More data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of IGF1RMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of JAK3More data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AlkMore data for this Ligand-Target Pair
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK2/cyclinAMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of INSRMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of FGFR3KMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ZAP70More data for this Ligand-Target Pair
TargetLysine--tRNA ligase(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of cMetMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Novartis Institute Of Biomedical Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKBalphaMore data for this Ligand-Target Pair