BindingDB PrimarySearch

Found 99 of ic50 for monomerid = 50536679

Ribosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Merck And

Curated by ChEMBL

IC50: <1nMAssay Description:Inhibition of full-length recombinant human His-tagged RPS6KA3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Testis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human His-tagged STK22D expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase TBK1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human GST-tagged TBK1 expressed in insect cells by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Tyrosine-protein kinase BTK(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: <1nMAssay Description:Inhibition of full-length recombinant human His-tagged BTK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 1.30nMAssay Description:Inhibition of full-length human His-tagged ABL1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Receptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 1.90nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic FLT3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Death-associated protein kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 1.90nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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MAP/microtubule affinity-regulating kinase 4(Mus musculus)
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2nMAssay Description:Inhibition of MARK4 in mouse cortical neurons assessed as inhibition of okadaic acid-induced tau phosphorylation at S262 residue preincubated for 15 ...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

PC cid PC sid

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Cyclin-dependent kinase 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.20nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.20nMAssay Description:Inhibition of full-length recombinant human His-tagged CHEK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Tyrosine-protein kinase HCK(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.80nMAssay Description:Inhibition of full-length human N-terminal GST-tagged HCK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Ephrin type-B receptor 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.90nMAssay Description:Inhibition of recombinant human GST-tagged cytoplasmic EPHB2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Ephrin type-A receptor 8(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 2.90nMAssay Description:Inhibition of recombinant human GST-tagged cytoplasmic EPHA8 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Proto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3nMAssay Description:Inhibition of full-length recombinant human His-tagged SRC expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Leucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.10nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.20nMAssay Description:Inhibition of full-length recombinant human GST-tagged DYRK1A expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Macrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.30nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic CSF1R expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Cytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.5nMAssay Description:Inhibition of full-length recombinant human His-tagged BMX expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Vascular endothelial growth factor receptor 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.5nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic KDR expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Tyrosine-protein kinase Lck(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 3.90nMAssay Description:Inhibition of full-length recombinant human His-tagged LCK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Cyclin-dependent kinase 7(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.10nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK7 expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

PC cid PC sid

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NUAK family SNF1-like kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.20nMAssay Description:Inhibition of full-length recombinant human His-tagged NUAK1 expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Cyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.40nMAssay Description:Inhibition of full-length recombinant human GST and His-tagged CDK5/P25 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar

PC cid PC sid

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5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 4.60nMAssay Description:Inhibition of full-length recombinant human GST and His-tagged AMPK alpha1/beta1/gamma1 expressed in baculovirus expression system by LanthaScreen as...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia GoogleScholar

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Misshapen-like kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 6nMAssay Description:Inhibition of recombinant human His-tagged MINK1 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase 26(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 6.30nMAssay Description:Inhibition of full-length recombinant human GST-tagged MST4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Inhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 7.10nMAssay Description:Inhibition of full-length recombinant human GST-tagged IKK-epsilon expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Ribosomal protein S6 kinase beta-1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 8nMAssay Description:Inhibition of full-length recombinant human GST-tagged RPS6KB1 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Interleukin-1 receptor-associated kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 9nMAssay Description:Inhibition of recombinant human GST-tagged IRAK1 (194 to 712 residues) catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Fibroblast growth factor receptor 2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 11nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic FGFR2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Cyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 12nMAssay Description:Inhibition of full-length recombinant human His-tagged CDK9/cyclin T1 expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar

PC cid PC sid

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NT-3 growth factor receptor(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 13nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic NTRK3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Dual specificity protein kinase CLK2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 14nMAssay Description:Inhibition of recombinant human GST-tagged CLK2 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
B.MOAD GoogleScholar

PC cid PC sid

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Rho-associated protein kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 17nMAssay Description:Inhibition of recombinant human GST-tagged ROCK1 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase B-raf(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 19nMAssay Description:Inhibition of full-length recombinant human GST-tagged BRAF expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 20nMAssay Description:Inhibition of full-length recombinant human His-tagged PDK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Ephrin type-A receptor 3(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 22nMAssay Description:Inhibition of recombinant human His-tagged cytoplasmic EPHA3 expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Interleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 23nMAssay Description:Inhibition of full-length recombinant human His-tagged IRAK4 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Glycogen synthase kinase-3 beta(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 23nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Serine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 24nMAssay Description:Inhibition of full-length recombinant human GST-tagged PAK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Serine/threonine-protein kinase Chk2(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 24nMAssay Description:Inhibition of full-length recombinant human His-tagged CHEK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Tyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 26nMAssay Description:Inhibition of full-length recombinant human GST-tagged ITK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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cAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 27nMAssay Description:Inhibition of recombinant human His-tagged PRKACA catalytic domain expressed in Escherichia coli by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Aurora kinase B(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 28nMAssay Description:Inhibition of full-length recombinant human His-tagged AURKB expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Tyrosine-protein kinase JAK3(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 33nMAssay Description:Inhibition of recombinant human GST-tagged JAK3 catalytic domain expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Protein kinase C iota type(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 37nMAssay Description:Inhibition of full-length recombinant human His-tagged PRKCI expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

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Mitogen-activated protein kinase 13(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 39nMAssay Description:Inhibition of full-length recombinant human His-tagged MAPK13 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Protein kinase C zeta type(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 40nMAssay Description:Inhibition of full-length recombinant human PRKCZ expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

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Glycogen synthase kinase-3 alpha(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 42nMAssay Description:Inhibition of full-length human GST-tagged GSK3A expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

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Tyrosine-protein kinase SYK(Homo sapiens (Human))
Merck And

Curated by ChEMBL

BDBM50536679(CHEMBL4568087)

IC50: 42nMAssay Description:Inhibition of full-length recombinant human N-terminal GST-tagged cytoplasmic SYK expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Displayed 1 to 50 (of 99 total ) | Next | Last >>

Filter my 99 hits

Targets 98▿
- Mitogen-activated protein kinase 8 2
- Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1 1
- Tyrosine-protein kinase JAK1 1
- Receptor tyrosine-protein kinase erbB-2 1
- Hepatocyte growth factor receptor 1
- Non-receptor tyrosine-protein kinase TYK2 1
- Serine/threonine-protein kinase B-raf 1
- Glycogen synthase kinase-3 alpha 1
- Glycogen synthase kinase-3 beta 1
- Serine/threonine-protein kinase Nek6 1
- Protein kinase C iota type 1
- NUAK family SNF1-like kinase 1 1
- Receptor-type tyrosine-protein kinase FLT3 1
- Serine/threonine-protein kinase Nek4 1
- Serine/threonine-protein kinase Nek2 1
- Sphingosine kinase 1 1
- Serine/threonine-protein kinase PAK 1 1
- Protein kinase C theta type 1
- Tyrosine-protein kinase JAK3 1
- Dual specificity mitogen-activated protein kinase kinase 1 1
- MAP/microtubule affinity-regulating kinase 4 1
- Tyrosine-protein kinase JAK2 1
- Dual specificity mitogen-activated protein kinase kinase 6 1
- Tyrosine-protein kinase ZAP-70 1
- Leucine-rich repeat serine/threonine-protein kinase 2 1
- Serine/threonine-protein kinase Sgk1 1
- Ephrin type-A receptor 3 1
- Tyrosine-protein kinase BTK 1
- Tyrosine-protein kinase ITK/TSK 1
- Insulin-like growth factor 1 receptor 1
- Epidermal growth factor receptor 1
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
- Ribosomal protein S6 kinase beta-1 1
- RAF proto-oncogene serine/threonine-protein kinase 1
- Serine/threonine-protein kinase 26 1
- Cyclin-dependent kinase 2 1
- Ephrin type-B receptor 2 1
- MAP kinase-activated protein kinase 2 1
- Ephrin type-A receptor 8 1
- MAP kinase-activated protein kinase 5 1
- Death-associated protein kinase 1 1
- PAS domain-containing serine/threonine-protein kinase 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
- Beta-adrenergic receptor kinase 1 1
- Cyclin-dependent kinase 7 1
- Serine/threonine-protein kinase pim-1 1
- Serine/threonine-protein kinase TAO2 1
- Testis-specific serine/threonine-protein kinase 1 1
- Angiopoietin-1 receptor 1
- Mast/stem cell growth factor receptor Kit 1
- Serine/threonine-protein kinase MRCK alpha 1
- Protein-tyrosine kinase 6 1
- Mitogen-activated protein kinase 14 1
- Activin receptor type-1B 1
- Casein kinase II subunit alpha 1
- Cyclin-dependent kinase 5 activator 1 1
- Interleukin-1 receptor-associated kinase 4 1
- Cytoplasmic tyrosine-protein kinase BMX 1
- RAC-gamma serine/threonine-protein kinase 1
- Interleukin-1 receptor-associated kinase 1 1
- Tyrosine-protein kinase ABL1 1
- RAC-alpha serine/threonine-protein kinase 1
- Rho-associated protein kinase 2 1
- Rho-associated protein kinase 1 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Mitogen-activated protein kinase 1 1
- 3-phosphoinositide-dependent protein kinase 1 1
- Tyrosine-protein kinase Lck 1
- NT-3 growth factor receptor 1
- Mitogen-activated protein kinase 9 1
- G protein-coupled receptor kinase 4 1
- Dual specificity protein kinase CLK2 1
- High affinity nerve growth factor receptor 1
- G protein-coupled receptor kinase 6 1
- Calcium/calmodulin-dependent protein kinase type IV 1
- Serine/threonine-protein kinase N1 1
- Tyrosine-protein kinase SYK 1
- Ribosomal protein S6 kinase alpha-3 1
- Serine/threonine-protein kinase TBK1 1
- Cyclin-T1/Cyclin-dependent kinase 9 1
- Aurora kinase B 1
- Vascular endothelial growth factor receptor 2 1
- Insulin receptor 1
- Tyrosine-protein kinase HCK 1
- Fibroblast growth factor receptor 2 1
- Serine/threonine-protein kinase PLK1 1
- Inhibitor of nuclear factor kappa-B kinase subunit beta 1
- Mitogen-activated protein kinase 13 1
- RAC-beta serine/threonine-protein kinase 1
- Casein kinase I isoform alpha 1
- Misshapen-like kinase 1 1
- Macrophage colony-stimulating factor 1 receptor 1
- cAMP-dependent protein kinase catalytic subunit alpha 1
- Protein kinase C zeta type 1
- Serine/threonine-protein kinase Chk2 1
- Serine/threonine-protein kinase Chk1 1
- SRSF protein kinase 1 1
Publications 1▿
- Bioorg Med Chem Lett 26: 4362-6 (2016) 99
Institutions 1▿
- Merck And 99
Affinity: 1 to 1.0E+4 nM▿
- IC50 99
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 0