TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 0.440nMAssay Description:Inhibition of ACE2 (unknown origin)More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 0.440nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 0.440nMAssay Description:This is a review article.More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:This is a review article.More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant human ACE2 using 7-Mca-YVADAPK (Dnp) as substrate by fluorescence plate reader assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 1.40nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of recombinant human ACE2 using 7-Mca-YVADAPK (Dnp) as substrate by fluorescence plate reader assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 4.20nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 expressed in HEK293T cells using FMZ as substrate by NanoLuc luciferase assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 expressed in HEK293T cells using FMZ as substrate by NanoLuc luciferase assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 9.80nMAssay Description:Inhibition of recombinant human ACE2 using 7-Mca-YVADAPK (Dnp) as substrate by fluorescence plate reader assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 expressed in HEK293T cells using FMZ as substrate by NanoLuc luciferase assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 expressed in HEK293T cells using FMZ as substrate by NanoLuc luciferase assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 expressed in HEK293T cells using FMZ as substrate by NanoLuc luciferase assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 21nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 expressed in HEK293T cells using FMZ as substrate by NanoLuc luciferase assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 32nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 52nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 76nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 by ITC assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 by ITC assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of SARS-COV2 S-RBD binding to human ACE2 by ITC assayMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:This is a review article.More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:This is a review article.More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 270nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 290nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 300nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 340nMpH: 6.5 T: 2°CAssay Description:Enzyme assay was conducted in 384-well microplates format. Activity was monitored by measuring increase in fluorescence (excitation @320 nm, emission...More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Functional H2 receptor antagonistic activity in vitro assay on the isolated spontaneously beating guinea-pig right atriumMore data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Ligand Info
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Affinity DataIC50: 5.47E+3nMAssay Description:This is a review article.More data for this Ligand-Target Pair
TargetAngiotensin-converting enzyme 2(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (Chuv) And University Of Lausanne (Unil
Curated by ChEMBL