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Found 15 Enz. Inhib. hit(s) with all data for entry = 50017174
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]neurotensin from human NTSR1 expressed in CHO cell membranes by radioligand depletion assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR1 F2.65C mutant expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR2 expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600200(CHEMBL5175252)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]neurotensin from human NTSR1 expressed in CHO cell membranes by radioligand depletion assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600200(CHEMBL5175252)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR2 expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600201(CHEMBL5184967)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR2 expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600199(CHEMBL5171551)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]neurotensin from human NTSR1 expressed in CHO cell membranes by radioligand depletion assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600201(CHEMBL5184967)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]neurotensin from human NTSR1 expressed in CHO cell membranes by radioligand depletion assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600199(CHEMBL5171551)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR1 F2.65C mutant expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600199(CHEMBL5171551)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR2 expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600198(CHEMBL5199274)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR1 F2.65C mutant expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600201(CHEMBL5184967)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR1 F2.65C mutant expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600198(CHEMBL5199274)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]neurotensin from human NTSR1 expressed in CHO cell membranes by radioligand depletion assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600200(CHEMBL5175252)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR1 F2.65C mutant expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg

Curated by ChEMBL
LigandPNGBDBM50600198(CHEMBL5199274)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR2 expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed