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Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50033877
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataKi:  760nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataKi:  760nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataKi:  880nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at rat recombinant TRPM8 receptor expressed in HEK293 cells assessed as inhibition of 0.25 uM icilin-induced stimulation of intra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataIC50:  710nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataIC50:  950nMAssay Description:Antagonist activity at rat recombinant TRPM8 receptor expressed in HEK293 cells assessed as inhibition of 0.25 uM icilin-induced stimulation of intra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataIC50:  1.20E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataIC50:  1.50E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataIC50:  2.30E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as inhibition of 0.1 um capsaicin-induced stimulation of intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataIC50:  3.27E+3nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataIC50:  3.46E+3nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as inhibition of 0.1 um capsaicin-induced stimulation of intracellular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataIC50:  1.30E+4nMAssay Description:Antagonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as inhibition of 100 uM allyl isothiocyanate-induced stimula...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataEC50:  700nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50318487(CHEMBL497318 | Cannabigerol)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed