Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50033877
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Antagonist activity at rat recombinant TRPM8 receptor expressed in HEK293 cells assessed as inhibition of 0.25 uM icilin-induced stimulation of intra...More data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Antagonist activity at rat recombinant TRPM8 receptor expressed in HEK293 cells assessed as inhibition of 0.25 uM icilin-induced stimulation of intra...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as inhibition of 0.1 um capsaicin-induced stimulation of intracellular...More data for this Ligand-Target Pair
Affinity DataIC50: 3.27E+3nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB1 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.46E+3nMAssay Description:Displacement of [3H]-CP-55,940 from human recombinant CB2 receptor expressed in HEK293 cells membrane incubated for 90 minsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Antagonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as inhibition of 0.1 um capsaicin-induced stimulation of intracellular...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as inhibition of 100 uM allyl isothiocyanate-induced stimula...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 4.40E+3nMAssay Description:Agonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fl...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Agonist activity at rat recombinant TRPV2 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita` Del Piemonte Orientale
Curated by ChEMBL
Universita` Del Piemonte Orientale
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at human TRPv1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dye based fl...More data for this Ligand-Target Pair